ECSOC-3 Conference Hall

ECSOC-3: http://www.mdpi.org/ecsoc-3.htm

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A. General Organic Synthesis

Dr. Thomas Wirth, Institut fuer Organische Chemie der Universitaet Basel, St. Johanns-Ring 19, CH-4056 Basel, Switzerland. Tel.: +41-61-267 1146 Fax: +41-61-267 1105, E-mail: [email protected]

[a0001] Cyclizations of 5,6-difunctionalized pyrido[2,3-d]pyrimidinetriones.
Wolfgang Stadlbauer and Dang Van Tinh.

[a0002] Influence of Some Thia or Azasubstituted Butyric Acid Derivatives on Chemical Shift of Carbon Atom of Benzene Ring.
Johannes Fröhlich, Sauter Fritz and Viktor Milata.

[a0003] Stereoselective a-Oxyfunctionalisation of Benzo(hetera)cyclanones by Dimethyldioxirane.
 Attila Kiss, József Jeko, Albert Lévai, Tamás Patonay.

[a0004] Indole, Cinnoline, Benzothiazine and Dihydrofuroquinoline Derivatives from Aryldifurylmethanes.
Alexander V. Butin, Vladimir T. Abaev, Tat'yana A. Stroganova, Andrey V. Gutnov, Irina V. Lodinaand Olga V. Shurakova.

[a0005] Symmetric Difuryl- and Trifurylmethanes: General Methods of Synthesis.
Tat'yana A. Stroganova, Alexander V. Butin, Lyudmila N. Sorotskaya and Vladimir G. Kul'nevich.

[a0006]Asymmetric Synthesis of Quaternary a-Amino Acids Using D-Ribonolactone Acetonide as a Chiral Auxiliary.
Marcial Moreno-Mañas, Elisenda Trepat, Rosa M. Sebastián and Adelina Vallribera.

[a0007] 1,3-Dipolar Cycloadditions of N-Benzyl Furfuryl Nitrones to Vinyl Ethers and a,b-Unsatureted Esters.
T. Tejero, S. Anoro, F.L. Merchan and P. Merino.

[a0008] Disulfonamides derived from camphor: A new ligand for the titanium alkoxide-promoted addition of diethylzinc to benzaldehyde.
Oscar Prieto, Diego J. Ramón and Miguel Yus.

[a0009] Sulfidation of  Heterocyclic 1,3-Dicarbonyl Systems .
Barbara Schnell and Thomas Kappe.

[a0010] The synthesis of g-hydroxy-a,b-unsaturated compounds from chiral cyanohydrins.
Jan Marcus, Johannes Brussee and Arne van der Gen.

[a0011] Synthesis of 4,5-dihydroimidazole-2-carboxamides.
V.N. Yarovenko, S.A. Kosarev, I.V. Zavarzin and M.M. Krayushkin.

[a0012] Isomeric Isoxazolopyridinones: Synthesis, Tautomerism and Molecular Orbital Calculation.
Robert Weis, Klaus Schweiger and Walter M. F. Fabian.

[a0013] The T1 Linker: Multidirectional Cleavage for Solid Phase Organic Synthesis.
Stefan Bräse, Stefan Dahmen and Matthias Lormann.

[a0014] A New Tungsten Complex Derived from [(Diphenylphosphino)methyl]diphenylphosphine oxide.
C. López-Leonardo, M. Alajarín, P. Llamas.

[a0015] New routes to dibenzobarrelene and pyrimidinobenzobarrelenes: a synthetic and computational study.
Mirta Golic, Douglas N. Butler, Ronald N. Warrener and Davor Margetic.

[a0016] Functionalised Rigid Rods - Dream or Reality.
Davor Margetic, Martin R. Johnston, Ronald N. Warrener.

[a0017] Site and Stereoselectivities in the High Pressure Reactionof Furan with Dimethyl 7-isopropylidenebicyclo[2.2.1]hepta-2,5-diene-2,3-dicarboxylate and Tetramethyl7-isopropylidenebicyclo[2.2.1]hepta-2,5-diene-2,3,5,6-tetracarboxylate.
Ronald N. Warrener, Douglas N. Butler, Shudong Wang and Edward R. T. Tiekink.

[a0018] Synthesis of Non-Racemic 1-Hydroxy Cycloalkenecarboxylic Acids by Metathesis of Dialkylated Glycolate Derivatives.
Liliana Parra Rapado, Vajira Bulugahapitiya and Philippe Renaud.

[a0019] Synthesis of Heterocycles Using Tandem Cyclization Processes.
Albert Padwa.

[a0020] N-Methyltyramine and N,O-Dimethyltyramine Synthesis via Intermediate 4-Methoxyphenyl-N-methyltioacetamide.
Vladimir N. Bulavka, Alexander N. Shchavlinskii and Oleg N. Tolkachev.

[a0021] 2-Methylbenzothiazole synthesis from 2-Mercaptoaniline and Acetic Acid.
Vladimir N. Bulavka, Tatiana N. Boiko and Igor I. Boiko.

[a0022] Microwave Enhanced Hydroamination of Styrene.
Julio A. Seijas, M. Pilar Vázquez Tato and M.Montserrat Martínez.

[a0023] Microwave Enhanced Synthesis of Quinazolines.
Julio A. Seijas, M. Pilar Vázquez Tato and M.Montserrat Martínez.

[a0024] Microwave Enhanced Knoevenagel Reaction: an expeditious method to prepare 3-benzylidene-1,3-dihydroindol-2-ones.
Julio A. Seijas, M. Pilar Vázquez Tato, M. Carmen Fernández and Nazaret Arias.

[a0025] Hydroamination of Cinnamyl Alcohol.
Julio A. Seijas, M. Pilar Vázquez-Tato, Luis Barreiro-Castro and Raquel Romero-Van-der-Schoot.

[a0026] Microwave promoted radical cyclization of trihaloacetamides.
Julio A. Seijas, M. Pilar Vázquez-Tato and Mercedes Jover.

[a0027] Synthesis of 3-benzylidene-1-methylpyrrolidin-2-one through 3-chloromethylene-1-methylpyrrolidin-2-one.
Julio A. Seijas, M. Pilar Vázquez-Tato, Luis Barreiro-Castro and Pablo Díaz.

[a0028] Dendrimeric Organic Reagents for Macromolecular Cross-Linking: Synthetic Approaches to 2,6-Bis[3,6-dioxa-9,9'-bis[bis[2-((p-carboxyphenoxy)carbonyl) ethyl]phosphinyl]nonyl] heptanedioic Acid [Bis(p-BCCEP-NHPDA)]].
Timothy A. Roach and Ramachandra S. Hosmane.

[a0029] A New Synthetic Approach toward Ring-Expanded ("Fat") Purine Nucleobases: Synthesis and Use of 5-Dichloromethyl-1-p-methoxybenzyl-4-nitroimidazole as a Versatile Intermediate.
Saika Siddiqui, Bruce Gustafson and Ramachandra S. Hosmane.

[a0030] Novel Imidazole Analogues of Stilbene: Synthesis and Characterization of Cis- and Trans-1,2-bis(4-nitro-1-p-methoxybenzylimidazol-5-yl)ethene.
Saika Siddiqui and Ramachandra S. Hosmane.

[a0031] Photochromic Fulgides: Transformation of Non-phtochromic (Z)-Isomer of a Fulgide into Highly Phtochromic (E)-Isomer via Structural Modification Containing Enhanced Conjugation.
Zhiyuan Sun and Ramachandra S. Hosmane.

[a0032] A Versatile Synthetic Precursor for Introduction of Specific N6-Modifications in 2,6-Diaminopurine Nucleosides:N2-Acetyl-2',3',5'-tri-O-acetyl-N6-(1,2,4-triazol-1-yl)- 2,6-diaminopurine-9--D-ribofuranoside.
XiaoHua Xu, Zhiyuan Sun and Ramachandra S. Hosmane.

[a0033] Base-Pairing Studies of a Ring-Expanded ("Fat") Nucleoside Analogue Possessing Potent Antiviral Activity.
Maria Bretner, Huanming Chen and Ramachandra S. Hosmane.

[a0034] Synthesis of Novel Acyclic Nucleoside and Acyclic Nucleoside Phosphonate Analogues of a Ring-Expanded ("Fat") Nucleobase Containing the Imidazo[4,5-e][1,3]diazepine Ring System.
Huanming Chen and Ramachandra S. Hosmane.

[a0035] A New, Improved Synthesis of 9-Benzyladenine: An Important Heterocyclic Analogue of Adenosine Useful for Chemical and Biochemical Research of Nucleic Acids.
Zhiyuan Sun and Ramachandra S. Hosmane.

[a0036] Titanocenes Catalyzed Diastereoselective Epoxidation of Allylic Alcohols.
Alessandra Lattanzi, Antonio Proto and Arrigo Scettri.

[a0037] A Novel Approach to the Synthesis of Substututed Indoles via Nitrilic Condensation.
G.B. Lapa and O.N. Tolkachev.

[a0038] Synthesis and Reactivity of 5-Functionalized 4-Hydroxyhexahydropyrimidine-2- thiones/ones.
Anatoly D. Shutalev.

[a0039] Phthalides and Chromones from 4-Coumarinacetic acids, Study of Beneficial Effects of Microwave Irradiation on Synthesis.
Margita Lacova, Dusan Loos, Jarmila Chovancova and Katarina Kralova.

[a0040] A New Route for the Synthesis of Cyclic Thioureas and Related Compounds.
Anatoly D. Shutalev.
 

B. Combinatorial Synthesis, Parallel Synthesis and Automation

Dr. Eduard Felder, Pharmaceuticals Division, Novartis, 4002 Basel, Switzerland. Tel.: +41 61 696 5293, Fax: +41 61 696 6174, E-mail: [email protected]

Dr. Andreas Marzinzik, Department of Chemistry BCC 315, The Scripps Research Institute, 10550 La Jolla, CA 92037, USA. Tel.: ++1 619-784-7515, Fax: ++1 619-784-7559, E-mail: [email protected]

[b0001] Colour Encoded Parallel Synthesis.
Lorenzo Williams.

[b0002] Polyhedral Oligosilsesquioxanes as Biological Scaffolds.
Kevin D. Wyndham and Frank J. Feher.

[b0003] Single bead FTIR in the optimization of solid-phase combinatorial organic syntheses.
Bing Yan.

[b0004] New Supports for Solid-Phase Organic Synthesis: Development of Cross-Linked Polytetrahydrofuran-Polystyrene Resins.
Patrick H. Toy, Patrick Garibay, Thomas Hoeg-Jensen and Kim D. Janda.

[b0005] Symmetric Building Blocks and Combinatorial Functional Group Transformation as Versatile Strategies in Combinatorial Chemistry.
Jörg Steffen Früchtel, Karin Pflugseder, and Hubert Gstach.

[b0006] Preliminary Results: The Development of a Continuous Flow Injection Microreactor For Organic Synthesis and Combinatorial Applications using Wittig Chemistry.
V. Skelton, G.M. Greenway, S.J. Haswell, D.O. Morgan, P. Styring, B.H. Warrington and S.Y.F. Wong.

[b0007] Exploiting Poly(ethylene glycol) as a Matrix for Liquid-Phase Organic Synthesis.
Frank Sieber, Paul Wentworth Jr. and Kim D. Janda.

[b0008] A Novel High-Speed Method for the Generation of 4-Aryldihydropyrimidine Compound Libraries Using a Microwave-Assisted Biginelli Condensation Protocol.
C. Oliver Kappe and Rajender S. Varma.

[b0009] Coupling of Phenols to 2-Chlorotrityl Resins under Non-basic Conditions.
Bernd Renneberg and Werner Breitenstein.

[b0010]Multi-step Split Synthesis on the TridentTM: Parallel Solution-Phase Synthesis of Urea and Amide Library.
Sukanta Bhattacharyya, Lisa Tamanaha, Lanchi Vo, Peter Wright and Jeff Labadie.

[b0011] Automation in Reaction Optimization.
Jay P. Chiang and K. Barry Sharpless.
 

C. Medicinal and Bioorganic Application of Organic Synthesis

Prof. Dr. Reinhard Neier, Institut de Chimie, Av. Bellevaux 51, CH-2000 Neuchatel, Switzerland. Tel.: +41 32 718 2428, Fax: +41 32 718 2511, E-mail: [email protected]

[c0001] Substrate Transport Limitation as tool to enhance enantioselectivity in the enzyme synthesis of chiral cyanohydrins.
Pieter Jan Gerrits, Johannes Brussee and Arne van der Gen.

[c0002] LQ12, A Novel PKC Activator, Enhances sAPP Secretion in PC-12 Cells.
Lixin Qiao, Rene Etcheberrigaray, Alan P. Kozikowski and Bryan Roth.

[c0003] A Novel Synthesis of Porphobilinogen: Synthetic and Biosynthetic Studies.
Reinhard Neier.

[c0004] Synthesis of N,N'-diarylalkanediamides and their antimycobacterial and antialgal activity.
L. Kubicova, K. Waisser, J. Kunesh, K. Kralova, S. Odlerova, M. Shlosarek, J. Janota and Z. Svoboda.

[c0005] Synthesis of some anilides of 2-alkylsulfanyl- and 2-chloro-6-alkylsulfanyl-4-pyridinecarboxylic acids and their photosynthesis-inhibiting activity .
Miroslav Miletin, Martin Dolezhal1, Jiri Hartl, Katarina Kralova and Milosh Machachek.

[c0006] Synthesis of Glycosyl Phosphoramidates: Novel Isosteric Analogs of Glycosyl Phosphates.
Thanukrishnan Kannan, Subramaniam Vinodhkumar and Duraikkannu Loganathan.

[c0007] Steroidal Tetraoxanes - New Class of Antitumor Compounds.
Dejan Opsenica, Gabriela Pocsfalvi, Zorica Juranic and Bogdan Solaja.

[c0008] A small company perspective on partnering with large pharma.
John W. Babich and Wendy A. Graham.

[c0009] Cold plasma induced chemical reactions. Implications for molecular evolution.
Constantin Romanescu and Cristofor I. Simionescu.
 
 

D. Natural Product Isolation and Modification

Prof. Dr. Atta-ur-Rahman and Dr. M. Iqbal Choudhary ( E-mails: [email protected]), H.E.J. Research Institute of Chemistry, University of Karachi, Karachi-75270, Pakistan. Tel.: +92-21-4990007 and 4986151, Fax: +92-21-4963124 and 4963373, E-mail: [email protected], URL: http://www.hej.edu.pk

[d0001] Stereoselective Synthesis of New Podophyllotoxin Derivative: 4-cyano-4-deoxy-4’- demethylepipodophyllotoxin.
Zai-Xin Chen, Wei-Yong Ma and Chun-Nian Zhang.

[d0002] Antifungal Activities and Essential Oil Constituents of Some Spices from Pakistan.
Atta-ur-Rahman, M.Iqbal Choudhary, Afgan Farooq, Aftab Ahmed, M. Zafar Iqbal, Betül Demirci, Fatih Demirci and K. Hüsnü Can Baser.
 

E. Information and Compound Archives Management and Internet Application

Dr. Shu-Kun Lin, Molecular Diversity Preservation International (MDPI), Saengergasse 25, CH-4054 Basel, Switzerland. Tel.: +41 79 322 3379, Fax: +41 61 302 8918, E-mail: [email protected]
Dr. Luc Patiny, Institute of Organic Chemistry, University Lausanne, ICO-BCH, 1015 Lausanne, Switzerland. Tel : +41 21 692 40 69 (Handy: +41 76 377 3110), Fax : +41 21 692 39 55, Email: [email protected]

[e0001] On the need for multiple lists of chemical information.
Jonathan Goodman.

[e0002] MarvinSketch and MarvinView: Molecule Applets for the World Wide Web.
Peter Csizmadia.

[e0003] JChem: Searching and Managing Structures using Web Browsers.
Ferenc Csizmadia and András Volford.

[e0004] JChemPaint - Using the Collaborative Forces of the Internet to Develop a Free Editor for 2D Chemical Structures.
Stefan Krause, Egon Willighagen and Christoph Steinbeck.

[e0005] Spectroscopy on-line.
E. Kleinpeter and St. Thomas.

[e0006] MolBank: First Fully Web-Based Publication of Chemical Reaction Data
Shu-Kun Lin and Luc Patiny


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Last change: 2 September 1999
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